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CAS:86044-76-0|Acetyl-(D-Trp1,D-Phe(4-Cl)2,D-Trp3,D-Arg6,D-Ala10)-LHRH|Ac-w-chloro-fwSYrLRPa-NH2

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ChinaPeptides Co., Ltd./强耀生物科技有限公司

NameAcetyl-(D-Trp1,D-Phe(4-Cl)2,D-Trp3,D-Arg6,D-Ala10)-LHRH
Code[86044-76-0]
The aliasAcetyl-(D-Trp1,D-Phe(4-Cl)2,D-Trp3,D-Arg6,D-Ala10)-LHRH
Sequence (single letter abbreviation)Ac-w-chloro-fwSYrLRPa-NH2
Sequence (three-letter abbreviation)Ac-D-Trp-4-chloro-D-Phe-D-Trp-Ser-Tyr-D-Arg-Leu-Arg-Pro-D-Ala-NH2(trifluoroacetate salt)
A basic descriptionAs a potent LHRH agonist, histrelin stimulates LH and FSH release and inhibits the actions of sex steroids on the male and female reproductive tracts. Its potency in vivo and in vitro is similar to that of the D-Trp6-containing analog. Especially because of its high water solubility and greater lipophilic character, histrelin appears promising for clinical application.Slow-release implants containing histreline implants were approved for the palliative treatment of advanced hormone-dependent prostate cancer.
solubility
The molecular weight1457.1
Chemical formulaC55H75N17O13
The purity80%，90%，95%，98%，99%
Weight1mg,5mg,10mg,50mg,100mg,1g
Storage conditionsStore at -20°C. Keep tightly closed. Store in a cool dry place.
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